Substance P/Neurokinin-1 Receptor Antagonist


Rolapitant Oral Tablet

Rolapitant may treat:

Rolapitant may prevent:

Rolapitant contraindicated conditions:

Rolapitant desired effects:

  • Decreased Brain Stem Substance P Activity
  • Emesis Suppression
  • Decreased Kinin Activity

Rolapitant drug classes:

  • Substance P/Neurokinin-1 Receptor Antagonist

Rolapitant pharmacologic actions:

  • Neurokinin-1 Receptor Antagonists

Rolapitant mechanism of action:

  • P-Glycoprotein Inhibitors
  • Breast Cancer Resistance Protein Inhibitors
  • Neurokinin 1 Antagonists
  • Cytochrome P450 2D6 Inhibitors
  • treatable

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Last updated: 10/19/2022, 7:14:13 AM